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作者:Cristiano Bolchi , Francesco Bavo , Marco Pallavicini
来源:[J].Amino Acids(IF 3.914), 2017, Vol.49 (5), pp.965-974
摘要:The enantiomers of amino acid benzyl esters are very important synthetic intermediates. Many of them are currently prepared by treatment with benzyl alcohol and p -toluenesulfonic acid in refluxing benzene or carbon tetrachloride, to azeotropically remove water, and then pre...
作者:... Simona Plutino , Sergio Fucile , Marco Pallavicini
来源:[J].European Journal of Medicinal Chemistry(IF 3.499), 2017, Vol.125, pp.1132-1144
摘要:Abstract(#br)Each of the four aromatic –CH= of ( S,R )-2-pyrrolidinyl-1,4-benzodioxane [( S,R )- 6 ] and of its epimer at the dioxane stereocenter ( S,S )- 6 , previously reported as α4β2 nAChR ligands, was replaced with nitrogen. The resulting four diastereoisomeric pairs o...
作者:Marco Pallavicini , Carlo Zanotto ...
来源:[J].European Journal of Medicinal Chemistry(IF 3.499), 2015, Vol.89, pp.252-265
摘要:Abstract(#br)A SAR study was performed on 3-substituted 2,6-difluorobenzamides, known inhibitors of the essential bacterial cell division protein FtsZ, through a series of modifications first of 2,6-difluoro-3-nonyloxybenzamide and then of its 3-pyridothiazolylmethoxy analogue PC...
作者:Marco Pallavicini , Giuseppe Chiodini ...
来源:[J].European Journal of Medicinal Chemistry(IF 3.499), 2016, Vol.120, pp.227-243
摘要:Abstract(#br)Lipophilic substituents at benzodioxane C (7) of 3-(benzodioxan-2-ylmethoxy)-2,6-difluorobenzamide improve the antibacterial activity against methicillin-resistant Staphylococcus aureus strains to MIC values in the range of 0.2–2.5 μg/mL, whereas hydrophilic sub...
作者:... Cristiano Bolchi , Francesco Bavo , Marco Pallavicini
来源:[J].Tetrahedron Letters(IF 2.397), 2016, Vol.57 (18), pp.2009-2011
摘要:Abstract(#br)Unlike the diastereomeric 1-phenylethylammonium salts, the diastereomeric N -1-phenylethylamides of ( S )- and ( R )-1,4-benzodioxane-2-carboxylic acid show significant differences in fusibility and solubility so as to be efficiently resolved by precipitation of the ...
作者:... Francesca Fasoli , Milena Moretti , Marco Pallavicini
来源:[J].Bioorganic & Medicinal Chemistry Letters(IF 2.338), 2016, Vol.26 (23), pp.5613-5617
摘要:Abstract(#br)A series of 3-nitrophenyl and 3-hydroxyphenyl ethers of ( S )- N -methylprolinol bearing bulky and lipophilic substituents at phenyl C5 were tested for affinity at α4β2 and α3β4 nAChRs. The two phenyl ethers 5-substituted with 6-hydroxy-1-hexynyl showed hig...
作者:Marco Pallavicini , Ermanno Valoti
来源:[J].Pharmacological Research(IF 4.346), 2016, Vol.103, pp.215-226
摘要:Abstract(#br)The progression of prostate cancer (PC) to a metastatic hormone refractory disease is the major contributor to the overall cancer mortality in men, mainly because the conventional therapies are generally ineffective at this stage. Thus, other therapeutic options...
作者:Marco Pallavicini , Ermanno Valoti ...
来源:[J].Tetrahedron: Asymmetry(IF 2.115), 2000, Vol.11 (9), pp.1957-1964
摘要:Abstract(#br)An insight into the mechanism of the highly efficient resolution of 1-phenylethylamine with enantiomerically pure isopropylideneglycerol hydrogen phthalate is provided by comparison of physicochemical and X-ray crystallographic data of the two diastereomeric salts fo...
作者:Marco Pallavicini
来源:[J].Nuclear Inst. and Methods in Physics Research, A(IF 1.142), 2003, Vol.502 (1), pp.155-157
摘要:Abstract(#br)The Euso project is now under Phase A study at the European Space Agency. If approved, it will mark the beginning of a new generation of experiments, devoted to the study of the extreme energy cosmic rays by looking at the earth atmosphere from space.

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