全部文献期刊会议图书|学者科研项目
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作者:Christian Jarry , El Mokhtar Essassi
来源:[J].Tetrahedron(IF 2.803), 2011, Vol.67 (12), pp.2279-2286
摘要:Abstract(#br)Condensation of 5(3)-amino-3(5)-arylpyrazoles with 4-hydroxy-6-methylpyran-2-one leads to 5,7-dimethyl-2-arylpyrazolo[1,5- a ]pyrimidines, 5-alkoxycarbonylmethyl-7-methyl-2-arylpyrazolo[1,5- a ]pyrimidines and their isomeric 7-alkoxycarbonylmethyl-5-methyl-2-arylpyra...
作者:... Jean-Michel Leger , Christian Jarry , Sylvain Routier
来源:[J].Tetrahedron Letters(IF 2.397), 2011, Vol.52 (41), pp.5224-5228
摘要:Abstract(#br)An efficient and original Ugi multicomponent reaction of aminopyridines and aminopyrimidines is reported. Starting from aminotetrazine 6 or 7 , an isocyanide and an ortho -carboxybenzaldehyde, tetrazinoimidazoisoquinolinones were isolated, after few minutes of microw...
作者:Christian Jarry , Stephane Massip ...
来源:[J].European Journal of Medicinal Chemistry(IF 3.499), 2014, Vol.82, pp.214-224
摘要:Abstract(#br)In this report, we describe the synthesis of a novel library of α7 nAChR ligands based on the modulation of the quinuclidine, quinazoline and tropane moieties. Spirane derivatives were newly synthesized under stereo specific 1,3 dipolar cylcoadditions. Only amid...
作者:Christian Jarry , Philippe Bernard ...
来源:[J].European Journal of Medicinal Chemistry(IF 3.499), 2014, Vol.84, pp.718-730
摘要:Abstract(#br)Synthesis and functionalization strategies of the imidazo[1,2- b ]pyrazole core were developed giving a rapid access to three series of novel imidazo[1,2- b ]pyrazole type derivatives: C-2/C-6/C-7 trisubstituted, C-2/C-3/C-6 tri(hetero)arylated and C-2/C-3/C-6/C...
作者:Christian Jarry , Saïd Lazar
来源:[J].Tetrahedron(IF 2.803), 2012, Vol.68 (25), pp.5018-5024
摘要:Abstract(#br)A novel and effective route for the synthesis of 2,4-disubstituted pyrido[2,3- d ]pyrimidines III is reported starting from the corresponding 2,4-dichloropyridopyrimidine 1 through regioselective functionalization palladium-catalyzed C–C coupling reactions, by t...
作者:... Isabelle Forfar-Bares , Jean-Jacques Bosc , Christian Jarry
来源:[J].Tetrahedron(IF 2.803), 2005, Vol.61 (18), pp.4453-4460
摘要:Abstract(#br)2-Substituted-4a-hydroxy-9 H -cycloalkyl[1,2- e ]oxazolo[3,2- a ]pyrimidin-9-ones 2a – c were synthesized by an one-step cyclocondensation from the 5-substituted-2-amino-2-oxazolines 1a – c with ethyl 2-oxocyclohexanecarboxylate in ethanol at room temperature, a...
作者:... Jean-Michel Léger , Christian Jarry , Jacques Robert
来源:[J].European Journal of Medicinal Chemistry(IF 3.499), 2012, Vol.54, pp.343-351
摘要:Abstract(#br)A series of mono- and bifunctional acyl compounds, build from the 8- O -azeloyl-14-benzoylaconine scaffold and differing by the length of the alkyl linker chain, were synthesised and evaluated against a panel of human tumour cell lines, A-549 (lung cancer), MCF-...
作者:... Thibaut Dupont , Christa E. Müller , Christian Jarry
来源:[J].Bioorganic & Medicinal Chemistry(IF 2.903), 2005, Vol.14 (8), pp.2697-2719
摘要:Abstract(#br)The development of potent and selective adenosine receptor ligands as potential drugs is an active area of research. Xanthines are one of the most important classes of adenosine receptor antagonists and have been widely developed in terms of affinity and selecti...
作者:Christian Jarry , El Mostapha Rakib ...
来源:[J].Tetrahedron(IF 2.803), 2005, Vol.61 (34), pp.8218-8225
摘要:Abstract(#br)In this paper, the synthesis of bi- and trisubstituted indazoles was described. 4-Alkoxy-7-aminoprotected-indazole or 7-aminoprotected-indazole derivatives were prepared selectively using SnCl 2 in alcohol or SnCl 2 in ethyl acetate, respectively. The effects of the ...
作者:... Philippe R Bovy , Christian Jarry , Sylvain Rault
来源:[J].Bioorganic & Medicinal Chemistry(IF 2.903), 2002, Vol.10 (4), pp.1043-1050
摘要:Abstract(#br)A series of trans,trans -1-phenyl-3-pyrrol-1-ylindan-2-carboxamide derivatives has been synthesized in eight steps starting from cinnamic acid or 3,3-diphenylpropionic acid. The trans,trans configuration of these carboxamides has been established by X-ray analysis an...

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